Over two days, the event will attract over 100 senior-level decision makers working in GPCR’s from the UK, Europe and US. This prestigious event will provide a forum for practitioners and prominent innovators to learn more about key solutions being provided to their industry, network with their peers, and address key industry concerns through a series of cutting edge conference presentations in a professional yet relaxed environment, during a 2 day conference programme.
Day 1
MEDICINAL CHEMISTRY
Focus upon the optimization of all areas of GPCR drug design including structure, mechanism, SAR, protein and ligand structure based drug design and molecular and in silico modelling
GPCR MODULATION
Closer studies into various aspects of GPCR’s including allosteric modulations from both a chemistry and biological aspect, dimerisation and oligomerisation.
Day 2
GPCR SCREENING
Examining the implementation of GPCR screening methods, HTS, HCS as well as exploring the roles of cell and label free screening, assay technology as well as determining cost effective assay formats.
GPCR SIGNALLING & DISCOVERY GPCR PROGRASMMES
Latest approaches to other important aspects of GPCR’s - including the role of signaling and trafficking, functional selectivity, polypharmacology and drug discovery programmes.
Event Agenda
